Investigational — Not Yet Approved

Cagrilintide

Phase 3 (REDEFINE program); Novo Nordisk filed an NDA for the combination product CagriSema (cagrilintide + semaglutide) in December 2025, FDA decision anticipated late 2026.

Cagrilintide is a long-acting synthetic amylin analogue that agonizes amylin (AMY1R/AMY3R) and calcitonin receptors, slowing gastric emptying and increasing satiety via hindbrain signaling. It is stud...

PubChem CID171397054
FormulaC194H312N54O59S2
Mol. Weight4409 g/mol

Sequence

Mechanism of Action

Cagrilintide is a long-acting synthetic amylin analogue that agonizes amylin (AMY1R/AMY3R) and calcitonin receptors, slowing gastric emptying and increasing satiety via hindbrain signaling. It is studied both alone and, more prominently, in combination with semaglutide, where it synergizes via complementary appetite pathways. In the Phase 3 REDEFINE 1 trial, the combination produced 20.4% mean weight reduction at 68 weeks versus 3.0% for placebo; gastrointestinal adverse events (nausea, vomiting, constipation) were the dominant safety finding, occurring in roughly 80% of combination-treated participants versus 40% on placebo, mostly mild-to-moderate.

Amylin receptor (AMY1R/AMY3R)Calcitonin receptor (CTR)

Research Literature